Bioactivity | D[LEU4,LYS8]-VP is a selective agonist of vasopressin V1b receptor, with the Kis of 0.16 nM, 0.52 nM, and 0.1.38 nM for rat, human and mouse V1b receptor, respectively. D[LEU4,LYS8]-VP has weak antidiuretic, vasopressor, and in vitro oxytocic activities[1][2]. |
Name | D[LEU4,LYS8]-VP |
CAS | 42061-33-6 |
Sequence | {Mpa}-Tyr-Phe-Leu-Asn-Cys-Pro-Lys-Gly (Disulfide bridge:Mpa1-Cys6) |
Shortening | {Mpa}-YFLNCPKG-NH2 (Disulfide bridge:Mpa1-Cys6) |
Formula | C47H67N11O11S2 |
Molar Mass | 1026.23 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |